Functional Groups
,
, Why studying functional groups is important
Histamine H1 antagonists
Challenges:
- Has low bioavailability 4% - bioavailability 80%
- Crosses bbb…..causes - Central nervous
drowsiness system-mediated
effect was suppressed
, Why studying functional groups is important
t1/2= 15 min
,
, Why studying functional groups is important
Histamine H1 antagonists
Challenges:
- Has low bioavailability 4% - bioavailability 80%
- Crosses bbb…..causes - Central nervous
drowsiness system-mediated
effect was suppressed
, Why studying functional groups is important
t1/2= 15 min